The biochemico-pharmacological tests showed that the combination of transplanted GABA receptors with [3H]GAEA could be inhibited by modullin, GABA agonist muscimol, GABA antagonists bicuculline and isopropyl bicyclophos phate.

• 移植GABA受体具有受体与配体结合的饱和特性,移植GABA受体与[~sH]GABA的结合可以被调变蛋白、蝇蕈醇、双可可碱及异丙基双环磷酸酯所抑制。