The transglycosylation process becomes potential targets for new antibiotics because of the remarkable ability of bacteria to develop resistance to antibiotics.

• 近年来，糖基转移酶的三维结构的确定，酶与抑制剂复合物结构及其相互作用的详细阐述，都为筛选和研究抑制糖基转移活性的新型抗生素提供了新的突破点。