The syntheses of some representative azole antifungals including ketoconazole, terconazole, itraconazole,posaconazole,fluconazole and voriconazole were reviewed.

• 对唑类抗真菌代表性药物酮康唑、特康唑、伊曲康唑、泊沙康唑、氟康唑和伏立康唑的主要合成方法进行了评述。