The previous studies indicated it produced anesthetic effect through its mimic GABA action ,which enhanced central inhibition mediated by postsynaptic GABAA receptors.

 
  • 近年来发现大多数全身麻醉药具有突触前效应,如抑制神经末梢突触前膜上的电压敏感性离子通道,从而引起突触前神经递质释放的改变:减少兴奋性神经递质释放或增加抑制性神经递质释放,最终抑制中枢突触传递。
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