Methods Starting from anisole,liarozole was synthesized by Friedel-Crafts(acylation,)nitration,nucleophilic substitution,reduction and cyclization.

 
  • 方法以苯甲醚为起始原料,经傅克酰基化、硝化、取代、还原、环合等7步反应得到目标化合物利阿唑。
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